Hamaguchi, Hisao; Amano, Yasushi; Moritomo, Ayako; Shirakami, Shohei; Nakajima, Yutaka et al. (2018). Discovery and structural characterization of peficitinib (ASP015K) as a novel and potent JAK inhibitor. Bioorganic and Medicinal Chemistry 26(18) , 4971-4983. 10.1016/j.bmc.2018.08.005. [PDB: 6aak] |
CMCF-ID |
Peer-Reviewed Article |
Health |
Heron, Paul W.; Abellán-Flos, Marta; Salmon, Laurent; Sygusch, Jurgen (2018). Bisphosphonate Inhibitors of Mammalian Glycolytic Aldolase. Journal of Medicinal Chemistry 61(23) , 10558-10572. 10.1021/acs.jmedchem.8b01000. [PDB: 5tle, 5tlh, 5tlw, 5tlz] |
CMCF-BM, CMCF-ID |
Peer-Reviewed Article |
Health |
Huguenin-Dezot, Nicolas; Alonzo, Diego A.; Heberlig, Graham W.; Mahesh, Mohan; Nguyen, Duy P. et al. (2018). Trapping biosynthetic acyl-enzyme intermediates with encoded 2,3-diaminopropionic acid. Nature 565(7737) , 112-117. 10.1038/s41586-018-0781-z. [PDB: 6ecb, 6ecc, 6ece, 6ecf] |
CMCF-ID |
Peer-Reviewed Article |
Health |
Ishiyama, N.; Ikura, M. (2018). Crystal structure of the alpha-E-catenin actin-binding domain. Protein Data Bank: 6dv1. |
CMCF-ID |
PDB Deposition |
Health |
Ishiyama, N.; Ikura, M. (2018). Crystal structure of the alpha-N-catenin actin-binding domain H1 mutant. Protein Data Bank: 6duy. |
CMCF-ID |
PDB Deposition |
Health |
Ishiyama, N.; Ikura, M. (2018). Crystal structure of the alpha-N-catenin actin-binding domain H1 mutant. Protein Data Bank: 6duw. |
CMCF-ID |
PDB Deposition |
Health |
Ishiyama, Noboru; Sarpal, Ritu; Wood, Megan N.; Barrick, Samantha K.; Nishikawa, Tadateru et al. (2018). Force-dependent allostery of the α-catenin actin-binding domain controls adherens junction dynamics and functions. Nature Communications 9(1) . 10.1038/s41467-018-07481-7. [PDB: 6duw, 6duy, 6dv1] |
CMCF-ID |
Peer-Reviewed Article |
Health |
Kundu, Prasun; Semesi, Anthony; Jore, Matthijs M.; Morin, Merribeth J.; Price, Virginia L. et al. (2018). Structural delineation of potent transmission-blocking epitope I on malaria antigen Pfs48/45. Nature Communications 9(1) . 10.1038/s41467-018-06742-9. [PDB: 6e62, 6e63, 6e64, 6e65] |
CMCF-ID |
Peer-Reviewed Article |
Health |
Kundu, P.; Semesi, A.; Julien, J.P. (2018). Crystal structure of malaria transmission-blocking antibody TB31F. Protein Data Bank: 6e65. |
CMCF-ID |
PDB Deposition |
Health |
Kundu, P.; Semesi, A.; Julien, J.P. (2018). Crystal structure of malaria transmission-blocking antibody 85RF45.1. Protein Data Bank: 6e64. |
CMCF-ID |
PDB Deposition |
Health |
Kundu, P.; Semesi, A.; Julien, J.P. (2018). Crystal structure of malaria transmission-blocking antigen Pfs48/45 6C in complex with antibody TB31F. Protein Data Bank: 6e63. |
CMCF-ID |
PDB Deposition |
Health |
Kundu, P.; Semesi, A.; Julien, J.P. (2018). Crystal structure of malaria transmission-blocking antigen Pfs48/45 6C in complex with antibody 85RF45.1. Protein Data Bank: 6e62. |
CMCF-ID |
PDB Deposition |
Health |
Loewen, P.C. (2018). B. pseudomallei KatG crystalized in the presence of ABTS. Protein Data Bank: 6mq1. |
CMCF-ID |
PDB Deposition |
Agriculture |
Loewen, P.C. (2018). B. pseudomallei KatG crystallized in the presence of furoyl hydrazide. Protein Data Bank: 6mq0. |
CMCF-ID |
PDB Deposition |
Agriculture |
Loewen, P.C. (2018). B. pseudomallei KatG crystallized in the presence of benzoyl hydrazide. Protein Data Bank: 6mpy. |
CMCF-ID |
PDB Deposition |
Agriculture |