Publication Beamlines Strategic Pillar
Kalliokoski, Tuomo; Kettunen, Henna; Kumpulainen, Esa; Kettunen, Emilia; Thieulin-Pardo, Gabriel et al. (2023). Discovery of novel methionine adenosyltransferase 2A (MAT2A) allosteric inhibitors by structure-based virtual screening. Bioorganic and Medicinal Chemistry Letters 94, 129450. 10.1016/j.bmcl.2023.129450. [PDB: 8p1t, 8p1v] CMCF-ID Health
Kattar, Solomon D.; Gulati, Anmol; Margrey, Kaila A.; Keylor, Mitchell H.; Ardolino, Michael et al. (2023). Discovery of MK-1468: A Potent, Kinome-Selective, Brain-Penetrant Amidoisoquinoline LRRK2 Inhibitor for the Potential Treatment of Parkinson’s Disease. Journal of Medicinal Chemistry . 10.1021/acs.jmedchem.3c01486. [PDB: 8six] CMCF-ID Health
Smith, Christopher R.; Chen, Dan; Christensen, James G.; Coulombe, René; Féthière, James et al. (2023). Discovery of Five SOS2 Fragment Hits with Binding Modes Determined by SOS2 X-Ray Cocrystallography. Journal of Medicinal Chemistry 67(1) , 774-781. 10.1021/acs.jmedchem.3c02140. [PDB: 8t5g, 8t5m, 8t5r] CMCF-BM, CMCF-ID Health
Thai, Elaine; Murugan, Rajagopal; Binter, Špela; Burn Aschner, Clare; Prieto, Katherine et al. (2023). Molecular determinants of cross-reactivity and potency by VH3-33 antibodies against the Plasmodium falciparum circumsporozoite protein. Cell Reports 42(11) , 113330. 10.1016/j.celrep.2023.113330. [PDB: 8fb5] CMCF-ID Health
Varkaris, Andreas; Pazolli, Ermira; Gunaydin, Hakan; Wang, Qi; Pierce, Levi et al. (2023). Discovery and clinical proof-of-concept of RLY-2608, a first-in-class mutant-selective allosteric PI3Ka inhibitor that decouples anti-tumor activity from hyperinsulinemia. Cancer Discovery . 10.1158/2159-8290.cd-23-0944. [PDB: 8ts7] CMCF-ID Health
Han Li; Dorothea Kominos; Jie Zhang; Alla Pritsker; Matthew Davison et al. (2023). Methods for treating inflammation using antibodies to kallidin and des-arg10-kallidin. Patent Number: US20230399388A1. CMCF-ID Health
Bailey-Elkin, B.A.; Mark, B.L. (2023). PRRSV-1 PLP2 domain. Protein Data Bank: 8ehn. CMCF-ID Health
Wang, F.; Cheng, W.; Yuan, Z.; Qi, J.; Li, J. et al. (2023). The Crystal Structure of integrase from Biortus. Protein Data Bank: 8wf7. CMCF-ID Health
Ali, Mohamed (2023). Investigating the role of acetylation of LC3-family proteins in regulating autophagy. Supervisor: Omichinski, James G.. Quebec, Canada: Université de Montréal. http://hdl.handle.net/1866/32170. CMCF-BM Health
Chadirji-Martinez, Kamil; Hudon, Guillaume; Chernikov, Roman; Heredia, Emillio; Feng, Renfei et al. (2023). Thorium speciation in ilmenite concentrates from the Mandena deposit, Madagascar: Implications for environmental remediation and thorium beneficiation. Applied Geochemistry , 105872. 10.1016/j.apgeochem.2023.105872. BIOXAS-SPECTROSCOPY, VESPERS Environment
Bartokova, Bibiana; Laredo, Thamara; Marangoni, Alejandro G.; Pensini, Erica (2023). Mechanism of tetrahydrofuran separation from water by stearic acid. Journal of Molecular Liquids 391, 123262. 10.1016/j.molliq.2023.123262. BXDS-WLE Environment
Bartokova, Bibiana; Marangoni, Alejandro G.; Laredo, Thamara; Pensini, Erica (2023). Effect of sorbitan ester structure on the separation between tetrahydrofuran and water. Frontiers in Soft Matter 3. 10.3389/frsfm.2023.1329058. BXDS-WLE, MID-IR Environment
Patel, Vedant; Marangoni, Alejandro G.; Ghazani, Saeed Mirzaee; Laredo, Thamara; Stobbs, Jarvis et al. (2023). Effect of bacterial surfactants on the phase behavior of miscible pollutants in water. Colloids and Surfaces C Environmental Aspects 1, 100013. 10.1016/j.colsuc.2023.100013. BXDS-WLE, MID-IR Environment
Jia, Xiaocen; Majzlan, Juraj; Ma, Liyuan; Liu, Peng; Fan, Peikuan et al. (2023). Novel insights into the mechanisms for Sb mobilization in groundwater in a mining area: A colloid field study. Journal of Hazardous Materials 459, 132212. 10.1016/j.jhazmat.2023.132212. CLS-APS Environment
Pastorek, Adam; Bernath, Peter; Boudon, Vincent (2023). High resolution infrared spectra of neopentane: Rovibrational analysis of bands at 8.3–6.4 μm. Journal of Quantitative Spectroscopy and Radiative Transfer 311, 108788. 10.1016/j.jqsrt.2023.108788. FAR-IR Environment