Sachdev Sidhu; Linda Beatty; Andreas Ernst (2012). Specific active site inhibitors of enzymes or substrate binding partners and methods of producing same. Patent Number: CA2807774A1. |
CMCF-ID |
Patent |
Health |
Sack, J. (2019). Crystal structure of RAR-related orphan receptor C (NHIS-RORGT(244-487)-L6-SRC1(678-692)) in complex with a phenyl (3-phenylpyrrolidin-3-yl)sulfone inhibitor. Protein Data Bank: 6p9f. |
CMCF-ID |
PDB Deposition |
Health |
Sack, John S.; Gao, Mian; Kiefer, Susan E.; Myers, Joseph E.; Newitt, John A. et al. (2016). Crystal structure of microtubule affinity-regulating kinase 4 catalytic domain in complex with a pyrazolopyrimidine inhibitor. Acta Crystallographica Section F:Structural Biology Communications 72(2) , 129-134. 10.1107/s2053230x15024747. [PDB: 5es1] |
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Peer-Reviewed Article |
Health |
Sack, J.S. (2020). SUBSTITUTED BENZYLOXYTRICYCLIC COMPOUNDS AS RETINOIC ACID-RELATED ORPHAN RECEPTOR GAMMA T AGONISTS. Protein Data Bank: 6xae. |
CMCF-ID |
PDB Deposition |
Health |
Sack, J.S. (2019). Crystal structure of JAK3 kinase domain in complex with a pyrrolopyridazine carboxamide inhibitor. Protein Data Bank: 6ny4. |
CMCF-ID |
PDB Deposition |
Health |
Sack, J.S. (2017). CRYSTAL STRUCTURE OF JAK3 KINASE DOMAIN IN COMPLEX WITH A PYRROLOPYRIDAZINE INHIBITOR. Protein Data Bank: 5vo6. |
CMCF-ID |
PDB Deposition |
Health |
Sack, J.S. (2015). CRYSTAL STRUCTURE OF MICROTUBULE AFFINITY-REGULATING KINASE 4 CATALYTIC DOMAIN IN COMPLEX WITH A PYRAZOLOPYRIMIDINE INHIBITOR. Protein Data Bank: 5es1. |
CMCF-ID |
PDB Deposition |
Health |
Sack, J.S. (2015). CRYSTAL STRUCTURE OF JANUS KINASE 2 IN COMPLEX WITH N,N-DICYCLOPROPYL-10-ETHYL-7-[(3-METHOXYPROPYL)AMINO] -3-METHYL-3,5,8,10-TETRAAZATRICYCLO[7.3.0.0,6] DODECA-1(9),2(6),4,7,11-PENTAENE-11-CARBOXAMIDE. Protein Data Bank: 5cf8. |
CMCF-ID |
PDB Deposition |
Health |
Sack, J.S. (2014). Crystal structure of JAK3 kinase domain in complex with a pyrrolopyridazine carboxamide inhibitor. Protein Data Bank: 4rio. |
CMCF-ID |
PDB Deposition |
Health |
Sack, J.S. (2011). Structure of Janus kinase 2 with a pyrrolotriazine inhibitor. Protein Data Bank: 3q32. |
CMCF-ID |
PDB Deposition |
Health |
Safaee, Nozhat; Kozlov, Guennadi; Noronha, Anne M.; Xie, Jingwei; Wilds, Christopher J. et al. (2012). Interdomain Allostery Promotes Assembly of the Poly(A) mRNA Complex with PABP and eIF4G. Molecular Cell 48(3) , 375-386. 10.1016/j.molcel.2012.09.001. [PDB: 4f02] |
CMCF-ID |
Peer-Reviewed Article |
Health |
Sahtout, Naheda; Kuttiyatveetil, Jijin R.A.; Sanders, David A.R. (2019). Structure and function of the putative thioredoxin 1 from the thermophilic eubacterium Thermosipho africanus strain TCF52B. Biochimica et Biophysica Acta - Proteins and Proteomics 1867(4) , 426-433. 10.1016/j.bbapap.2019.01.011. [PDB: 6mos] |
CMCF-ID |
Peer-Reviewed Article |
Health |
Sahtout, N.; Kuttiyatveetil, J.R.A.; Sanders, D.A.R. (2021). Structure of thioredoxin reductase from the thermophilic eubacterium Thermosipho africanus TCF52B. Protein Data Bank: 7jyp. |
CMCF-ID |
PDB Deposition |
Health |
Sakurada, I.; Endo, T.; Hikita, K.; Hirabayashi, T.; Hosaka, Y. et al. (2017). Discovery of novel aminobenzisoxazole derivatives as orally available factor IXa inhibitors. Protein Data Bank: 5tnt. |
CMCF-ID |
PDB Deposition |
Health |
Sakurada, Isao; Endo, Toshiya; Hikita, Katsuyoshi; Hirabayashi, Tomokazu; Hosaka, Yoshitaka et al. (2017). Discovery of novel aminobenzisoxazole derivatives as orally available factor IXa inhibitors. Bioorganic and Medicinal Chemistry Letters 27(11) , 2622-2628. 10.1016/j.bmcl.2017.03.002. [PDB: 5tnt] |
CMCF-ID |
Peer-Reviewed Article |
Health |